Minoxidil was originally developed as a blood pressure medication; once its hair-growth side effect was noticed, it was reformulated topically (and later as low-dose oral) for hair loss.

Mechanism of Action

The exact mechanism is still being studied, but it's believed to increase blood flow to follicles and modulate growth factors in ways that prolong the anagen phase and encourage follicles to shift to a larger diameter.

Use and Efficacy

Topical 5% solution/foam is applied once or twice daily. Low-dose oral minoxidil (0.25-5 mg/day) is increasingly favored, especially for patients who don't respond to or struggle with the topical form; in efficacy rankings it falls behind dutasteride and finasteride.

Side Effects

The most common topical side effects are contact dermatitis and unwanted hair growth elsewhere (hypertrichosis). Oral use can cause dose-dependent hypertrichosis and cardiovascular effects (palpitations, fluid retention).

Relevance to transplantation: Minoxidil is not a substitute for surgery โ€” it helps slow loss of existing, DHT-sensitive follicles. Many surgeons recommend continuing it after transplant surgery to protect non-transplanted native hair.